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PLX4720

Synonyms

SourcesNames Used
CCLE, GDSC1000PLX4720
CTRPv2PLX-4720
PharmacoGx PLX4720

External IDs

DatabaseIdentifier
Smiles: CCCS(=O)(=O)NC1=C(C(=C(C=C1)F)C(=O)C2=CNC3=NC=C(C=C23)Cl)F
Inchikey: YZDJQTHVDDOVHR-UHFFFAOYSA-N
Pubchem: 24180719

Annotated Targets

BRAF, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to PLX4720


Feature TypeStandardized
Nominal ANOVA
mRNA IKZF1 CCLE pan-cancer AAC -0.39 4e-05
mRNA ARHGAP30 CCLE pan-cancer AAC -0.36 5e-05
mRNA CD53 CCLE pan-cancer AAC -0.33 0.0003
mRNA MAP4K1 CCLE pan-cancer AAC -0.31 2e-05
mRNA MFNG CCLE pan-cancer AAC -0.3 4e-05
mRNA KLHL6 CCLE pan-cancer AAC -0.28 0.0003
mRNA ARHGAP30 GDSC1000 pan-cancer AAC -0.26 0.0001
mRNA CCDC88C CCLE pan-cancer AAC -0.26 1e-05
mRNA WAS CCLE pan-cancer AAC -0.26 0.0006
mRNA LRMP CCLE pan-cancer AAC -0.25 0.0002
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