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PLX4720

Synonyms

SourcesNames Used
CCLE, GDSC1000PLX4720
CTRPv2PLX-4720
PharmacoGx PLX4720

External IDs

DatabaseIdentifier
Smiles: CCCS(=O)(=O)NC1=C(C(=C(C=C1)F)C(=O)C2=CNC3=NC=C(C=C23)Cl)F
Inchikey: YZDJQTHVDDOVHR-UHFFFAOYSA-N
Pubchem: 24180719

Annotated Targets

BRAF, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to PLX4720


Feature TypeStandardized
Nominal ANOVA
mRNA ICAM2 CCLE pan-cancer AAC -0.22 0.0001
mRNA IL2RG CCLE pan-cancer AAC -0.21 0.002
mRNA ATP8A1 CCLE pan-cancer AAC -0.21 6e-05
mRNA SEPT1 CCLE pan-cancer AAC -0.21 0.0003
mRNA PIK3CG CCLE pan-cancer AAC -0.21 0.003
mRNA RASSF5 CCLE pan-cancer AAC -0.21 0.002
mRNA INPP5B CCLE pan-cancer AAC -0.21 0.0003
mRNA PPP1R16B CCLE pan-cancer AAC -0.21 0.0007
mRNA RASAL3 CCLE pan-cancer AAC -0.21 0.002
mRNA RAD17 CCLE pan-cancer AAC -0.2 8e-05
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