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PLX4720

Synonyms

SourcesNames Used
CCLE, GDSC1000PLX4720
CTRPv2PLX-4720
PharmacoGx PLX4720

External IDs

DatabaseIdentifier
Smiles: CCCS(=O)(=O)NC1=C(C(=C(C=C1)F)C(=O)C2=CNC3=NC=C(C=C23)Cl)F
Inchikey: YZDJQTHVDDOVHR-UHFFFAOYSA-N
Pubchem: 24180719

Annotated Targets

BRAF, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to PLX4720


Feature TypeStandardized
Nominal ANOVA
mRNA C10orf90 CCLE pan-cancer AAC 0.4 3e-09
mRNA INPP5F CTRPv2 pan-cancer AAC 0.41 5e-19
mRNA DCT CCLE pan-cancer AAC 0.42 8e-12
mRNA SOX10 CTRPv2 pan-cancer AAC 0.44 3e-15
mRNA SOX10 CCLE pan-cancer AAC 0.45 1e-09
mRNA ROPN1 CCLE pan-cancer AAC 0.47 2e-14
mRNA RXRG CCLE pan-cancer AAC 0.49 2e-17
mRNA TRIM51 CCLE pan-cancer AAC 0.5 1e-15
mRNA S100B CCLE pan-cancer AAC 0.51 1e-12
mRNA PLP1 CCLE pan-cancer AAC 0.56 8e-14
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