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VX-702

Synonyms

SourcesNames Used
GDSC1000VX-702
PharmacoGx VX-702

External IDs

DatabaseIdentifier
Smiles: C1=CC(=C(C(=C1)F)N(C2=NC(=C(C=C2)C(=O)N)C3=C(C=C(C=C3)F)F)C(=O)N)F
Inchikey: FYSRKRZDBHOFAY-UHFFFAOYSA-N
Pubchem: 10341154

Annotated Targets

MAPK11, MAPK12, MAPK14, TNF, IL1B, IL6

FDA Approval Status

Not Approved
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Top molecular features associated with response to VX-702


Feature TypeStandardized
Nominal ANOVA
mRNA LYL1 GDSC1000 pan-cancer AAC 0.15 0.004
mRNA SPAST GDSC1000 pan-cancer AAC 0.15 9e-05
mRNA POLG2 GDSC1000 pan-cancer AAC 0.15 8e-05
mRNA C16orf54 GDSC1000 pan-cancer AAC 0.16 0.0005
mRNA RNASE6 GDSC1000 pan-cancer AAC 0.16 3e-05
mRNA NPW GDSC1000 pan-cancer AAC 0.17 3e-06
mRNA NNAT GDSC1000 pan-cancer AAC 0.18 3e-07
mRNA ZNF407 GDSC1000 pan-cancer AAC 0.19 8e-07
mRNA MFNG GDSC1000 pan-cancer AAC 0.19 0.003
mRNA GUCA2B GDSC1000 pan-cancer AAC 0.19 2e-08
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