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SB 216763

Synonyms

SourcesNames Used
GDSC1000SB 216763
PharmacoGx SB 216763

External IDs

DatabaseIdentifier
Smiles: Cn1cc(C2=C(C(=O)NC2=O)c3ccc(Cl)cc3Cl)c4ccccc14
Pubchem: 176158

Annotated Targets

CCNA2, CDK2, GSK3A, GSK3B

FDA Approval Status

Not Approved
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Top molecular features associated with response to SB 216763


Feature TypeStandardized
Nominal ANOVA
mRNA ENSA GDSC1000 pan-cancer AAC -0.15 0.0002
mRNA SMAD9 GDSC1000 pan-cancer AAC -0.16 0.0002
mRNA IL7R GDSC1000 pan-cancer AAC 0.14 0.0002
mRNA TSPAN4 GDSC1000 pan-cancer AAC 0.17 0.0002
mRNA DKK1 GDSC1000 pan-cancer AAC 0.16 0.0002
mRNA SLC6A5 GDSC1000 pan-cancer AAC -0.14 0.0003
mRNA PHF8 GDSC1000 pan-cancer AAC -0.15 0.0003
mRNA C15orf52 GDSC1000 pan-cancer AAC 0.16 0.0003
mRNA ASH1L GDSC1000 pan-cancer AAC -0.14 0.0003
mRNA MAP4K4 GDSC1000 pan-cancer AAC 0.14 0.0004
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