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RDEA119

Synonyms

SourcesNames Used
GDSC1000RDEA119
FIMMRefametinib
PharmacoGx RDEA119

External IDs

DatabaseIdentifier
Smiles: COC1=CC(=C(C(=C1NS(=O)(=O)C2(CC2)CC(CO)O)NC3=C(C=C(C=C3)I)F)F)F
Inchikey: RDSACQWTXKSHJT-NSHDSACASA-N
Pubchem: 44182295

FDA Approval Status

Not Approved
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Top molecular features associated with response to RDEA119


Feature TypeStandardized
Nominal ANOVA
mRNA APLNR FIMM pan-cancer AAC -0.6 6e-05
mRNA IKZF1 GDSC1000 pan-cancer AAC -0.33 5e-06
mRNA RAB39B GDSC1000 pan-cancer AAC -0.29 7e-18
mRNA EML5 GDSC1000 pan-cancer AAC -0.29 1e-13
mRNA MAP4K1 GDSC1000 pan-cancer AAC -0.28 5e-10
mRNA RHOH GDSC1000 pan-cancer AAC -0.28 6e-09
mRNA MZB1 GDSC1000 pan-cancer AAC -0.27 8e-10
mRNA PHOX2A GDSC1000 pan-cancer AAC -0.27 1e-05
mRNA SEPT1 GDSC1000 pan-cancer AAC -0.27 1e-11
mRNA SBK1 GDSC1000 pan-cancer AAC -0.27 4e-15
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