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RDEA119

Synonyms

SourcesNames Used
GDSC1000RDEA119
FIMMRefametinib
PharmacoGx RDEA119

External IDs

DatabaseIdentifier
Smiles: COC1=CC(=C(C(=C1NS(=O)(=O)C2(CC2)CC(CO)O)NC3=C(C=C(C=C3)I)F)F)F
Inchikey: RDSACQWTXKSHJT-NSHDSACASA-N
Pubchem: 44182295

FDA Approval Status

Not Approved
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Top molecular features associated with response to RDEA119


Feature TypeStandardized
Nominal ANOVA
mRNA HEXB GDSC1000 pan-cancer AAC 0.29 6e-17
mRNA DUSP6 GDSC1000 pan-cancer AAC 0.26 2e-16
mRNA GKAP1 GDSC1000 pan-cancer AAC -0.27 2e-16
mRNA TOR4A GDSC1000 pan-cancer AAC 0.28 2e-16
mRNA TSPO GDSC1000 pan-cancer AAC 0.27 6e-16
mRNA CD68 GDSC1000 pan-cancer AAC 0.26 6e-16
mRNA SERPINB1 GDSC1000 pan-cancer AAC 0.26 9e-16
mRNA CD63 GDSC1000 pan-cancer AAC 0.31 1e-15
mRNA CASP4 GDSC1000 pan-cancer AAC 0.25 1e-15
mRNA FNDC3B GDSC1000 pan-cancer AAC 0.26 1e-15
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