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RDEA119

Synonyms

SourcesNames Used
GDSC1000RDEA119
FIMMRefametinib
PharmacoGx RDEA119

External IDs

DatabaseIdentifier
Smiles: COC1=CC(=C(C(=C1NS(=O)(=O)C2(CC2)CC(CO)O)NC3=C(C=C(C=C3)I)F)F)F
Inchikey: RDSACQWTXKSHJT-NSHDSACASA-N
Pubchem: 44182295

FDA Approval Status

Not Approved
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Top molecular features associated with response to RDEA119


Feature TypeStandardized
Nominal ANOVA
mRNA ACVR1 GDSC1000 pan-cancer AAC 0.16 4e-06
mRNA ACYP1 GDSC1000 pan-cancer AAC -0.13 3e-05
mRNA ADAM10 GDSC1000 pan-cancer AAC 0.13 3e-05
mRNA ADAM9 GDSC1000 pan-cancer AAC 0.26 7e-11
mRNA ADCY7 GDSC1000 pan-cancer AAC 0.16 9e-07
mRNA ADGRB3 GDSC1000 pan-cancer AAC -0.17 8e-07
mRNA ADGRE2 GDSC1000 pan-cancer AAC 0.15 3e-06
mRNA ADGRE5 GDSC1000 pan-cancer AAC 0.24 1e-13
mRNA ADGRG6 GDSC1000 pan-cancer AAC 0.16 4e-06
mRNA ADGRL1 GDSC1000 pan-cancer AAC -0.16 4e-06
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