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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA ZYG11B CTRPv2 pan-cancer AAC -0.14 0.0001
mRNA ZSWIM5 CTRPv2 pan-cancer AAC -0.16 2e-05
mRNA ZSCAN26 CTRPv2 pan-cancer AAC -0.13 0.0002
mRNA ZNRF2 CCLE pan-cancer AAC 0.2 4e-05
mRNA ZNF81 CTRPv2 pan-cancer AAC -0.16 4e-06
mRNA ZNF791 CTRPv2 pan-cancer AAC -0.14 6e-05
mRNA ZNF775 gCSI pan-cancer AAC -0.25 4e-05
mRNA ZNF775 CTRPv2 pan-cancer AAC -0.17 7e-06
mRNA ZNF764 CTRPv2 pan-cancer AAC -0.16 8e-06
mRNA ZNF750 CCLE pan-cancer AAC 0.19 0.0001
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