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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA ABCA12 CCLE pan-cancer AAC 0.25 1e-07
mRNA ABCA12 gCSI pan-cancer AAC 0.24 4e-05
mRNA ABCA12 CTRPv2 pan-cancer AAC 0.14 0.0001
mRNA ABCC3 CCLE pan-cancer AAC 0.26 1e-06
mRNA ABCC3 GDSC1000 pan-cancer AAC 0.27 3e-06
mRNA ABCC6 GDSC1000 pan-cancer AAC 0.18 0.0002
mRNA ABI2 CCLE pan-cancer AAC -0.22 9e-06
mRNA ABTB2 CTRPv2 pan-cancer AAC 0.13 0.0002
mRNA ABTB2 gCSI pan-cancer AAC 0.25 0.0003
mRNA AC002310.13 CTRPv2 pan-cancer AAC -0.13 0.0003
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