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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA DUSP1 FIMM pan-cancer AAC -0.84 0.0003
mRNA NOX1 UHNBreast pan-cancer AAC -0.83 0.0002
mRNA NRBF2 FIMM pan-cancer AAC -0.7 0.0003
mRNA STX2 CCLE pan-cancer AAC -0.36 9e-13
mRNA IFFO1 CCLE pan-cancer AAC -0.35 3e-06
mRNA FAM216A CCLE pan-cancer AAC -0.33 5e-12
mRNA ZEB1 CCLE pan-cancer AAC -0.32 8e-11
mRNA LIX1L CCLE pan-cancer AAC -0.32 9e-10
mRNA PDZRN3 gCSI pan-cancer AAC -0.32 1e-06
mRNA CNRIP1 CCLE pan-cancer AAC -0.31 1e-07
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