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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA SCN7A FIMM pan-cancer AAC 0.69 1e-06
mRNA CORIN FIMM pan-cancer AAC 0.7 1e-06
mRNA C14orf105 FIMM pan-cancer AAC 0.72 5e-07
mRNA EPHA3 FIMM pan-cancer AAC 0.73 2e-07
mRNA CLUL1 FIMM pan-cancer AAC 0.76 2e-08
mRNA KCNJ13 FIMM pan-cancer AAC 0.77 2e-08
mRNA NUFIP1 UHNBreast pan-cancer AAC 0.82 0.0004
mRNA MYZAP UHNBreast pan-cancer AAC 0.83 0.0002
mRNA TNNC1 UHNBreast pan-cancer AAC 0.83 0.0002
mRNA N4BP2L2 UHNBreast pan-cancer AAC 0.93 2e-06
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