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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA DPP4 FIMM pan-cancer AAC 0.63 0.0003
mRNA COBLL1 FIMM pan-cancer AAC 0.63 6e-05
mRNA SCIN FIMM pan-cancer AAC 0.64 1e-05
mRNA CALCRL FIMM pan-cancer AAC 0.65 8e-06
mRNA KCNJ16 FIMM pan-cancer AAC 0.66 2e-05
mRNA SEMA3D FIMM pan-cancer AAC 0.66 4e-06
mRNA SPTBN2 FIMM pan-cancer AAC 0.67 2e-05
mRNA DLX6 FIMM pan-cancer AAC 0.68 4e-06
mRNA PPP1R1A FIMM pan-cancer AAC 0.68 1e-06
mRNA PDK4 FIMM pan-cancer AAC 0.69 8e-06
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